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@ARTICLE{Qiao:471682,
author = {Qiao, Jingxin and Li, Yue-Shan and Zeng, Rui and Liu,
Feng-Liang and Luo, Rong-Hua and Huang, Chong and Wang,
Yi-Fei and Zhang, Jie and Quan, Baoxue and Shen, Chenjian
and Mao, Xin and Liu, Xinlei and Sun, Weining and Yang, Wei
and Ni, Xincheng and Wang, Kai and Xu, Ling and Duan, Zi-Lei
and Zou, Qing-Cui and Zhang, Hai-Lin and Qu, Wang and Long,
Yang-Hao-Peng and Li, Ming-Hua and Yang, Rui-Cheng and Liu,
Xiaolong and You, Jing and Zhou, Yangli and Yao, Rui and Li,
Wen-Pei and Liu, Jing-Ming and Chen, Pei and Liu, Yang and
Lin, Gui-Feng and Yang, Xin and Zou, Jun and Li, Linli and
Hu, Yiguo and Lu, Guang-Wen and Li, Wei-Min and Wei, Yu-Quan
and Zheng, Yong-Tang and Lei, Jian and Yang, Shengyong},
title = {{SARS}-{C}o{V}-2 {M} pro inhibitors with antiviral activity
in a transgenic mouse model},
journal = {Science},
volume = {371},
number = {6536},
issn = {0036-8075},
address = {Cambridge, Mass.},
publisher = {Moses King},
reportid = {PUBDB-2021-04550},
pages = {1374 - 1378},
year = {2021},
abstract = {Vaccines are an important tool in the fight against
COVID-19, but developing antiviral drugs is also a high
priority, especially with the rise of variants that may
partially evade vaccines. The viral protein main protease is
required for cleaving precursor polyproteins into functional
viral proteins. This essential function makes it a key drug
target. Qiao et al. designed 32 inhibitors based on either
boceprevir or telaprevir, both of which are protease
inhibitors approved to treat hepatitis C virus. Six
compounds protected cells from viral infection with high
potency, and two of these were selected for in vivo studies
based on pharmokinetic experiments. Both showed strong
antiviral activity in a mouse model.},
cin = {DOOR ; HAS-User},
ddc = {500},
cid = {I:(DE-H253)HAS-User-20120731},
pnm = {6G3 - PETRA III (DESY) (POF4-6G3)},
pid = {G:(DE-HGF)POF4-6G3},
experiment = {EXP:(DE-H253)P-P11-20150101},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:33602867},
UT = {WOS:000636043400052},
doi = {10.1126/science.abf1611},
url = {https://bib-pubdb1.desy.de/record/471682},
}