% IMPORTANT: The following is UTF-8 encoded. This means that in the presence
% of non-ASCII characters, it will not work with BibTeX 0.99 or older.
% Instead, you should use an up-to-date BibTeX implementation like “bibtex8” or
% “biber”.
@ARTICLE{Meyer:82180,
author = {Meyer, U. and Bisel, P. and Weckert, E. and Frahm, A. W.
and DESY},
title = {{B}icyclic glutamic acid derivatives},
journal = {Chirality},
volume = {18},
issn = {0899-0042},
address = {New York, NY [u.a.]},
publisher = {Wiley Interscience},
reportid = {PHPPUBDB-4925},
pages = {394},
year = {2006},
abstract = {For the second-generation asymmetric synthesis of the
trans-tris(homoglutamic) acids via Strecker reaction of
chiral ketimines, the cyanide addition as the key
stereodifferentiating step produces mixtures of
diastereomeric alpha-amino nitrile esters the composition of
which is independent of the reaction temperature and the
type of the solvent, respectively. The subsequent hydrolysis
is exclusively achieved with concentrated H(2)SO(4) yielding
diastereomeric mixtures of three secondary alpha-amino
alpha-carbamoyl-gamma-esters and two diastereomeric
cis-fused angular alpha-carbamoyl gamma-lactams as bicyclic
glutamic acid derivatives, gained from in situ stereomer
differentiating cyclisation of the secondary cis-alpha-amino
alpha-carbamoyl-gamma-esters. Separation was achieved by CC.
The pure secondary trans-alpha-amino
alpha-carbamoyl-gamma-esters cyclise on heating and
treatment with concentrated H(2)SO(4), respectively, to
diastereomeric cis-fused angular secondary alpha-amino
imides. Their hydrogenolysis led to the enantiomeric
cis-fused angular primary alpha-amino imides. The
configuration of all compounds was completely established by
NMR methods, CD-spectra, and by X-ray analyses of the
(alphaR,1R,5R)-1-carbamoyl-2-(1-phenylethyl)-2-azabicyclo[3.3.0]octan-3-one
and of the
trans-alphaS,1S,2R-2-ethoxycarbonylmethyl-1-(1-phenylethylamino)cyclopentanecarboxamide.},
keywords = {Amino Acids, Cyclic: chemistry / Amino Acids, Cyclic:
metabolism / Circular Dichroism / Crystallography, X-Ray /
Cyclization / Esters: chemistry / Glutamic Acid: analogs
$\&$ derivatives / Glutamic Acid: chemistry / Hot
Temperature / Hydrolysis / Models, Chemical / Molecular
Structure / Nuclear Magnetic Resonance, Biomolecular /
Solvents: chemistry / Stereoisomerism / Sulfuric Acids:
pharmacology / Amino Acids, Cyclic (NLM Chemicals) / Esters
(NLM Chemicals) / Solvents (NLM Chemicals) / Sulfuric Acids
(NLM Chemicals) / Glutamic Acid (NLM Chemicals) / sulfuric
acid (NLM Chemicals)},
cin = {HASYLAB},
ddc = {570},
cid = {$I:(DE-H253)HASYLAB_-2012_-20130307$},
pnm = {Facility (machine) DORIS/PETRA (POF1-DORIS-PETRA-20130405)},
pid = {G:(DE-H253)POF1-DORIS-PETRA-20130405},
experiment = {EXP:(DE-H253)DORISIII(machine)-20150101},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:16596563},
UT = {WOS:000237279100010},
doi = {10.1002/chir.20260},
url = {https://bib-pubdb1.desy.de/record/82180},
}