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@ARTICLE{Graewert:618954,
author = {Graewert, Melissa A. and Volkova, Maria and Jonasson, Klara
and Määttä, Juha A. E. and Gräwert, Tobias and Mamidi,
Samara and Kulesskaya, Natalia and Evenäs, Johan and
Johnsson, Richard E. and Svergun, Dmitri and Bhattacharjee,
Arnab and Huttunen, Henri J.},
title = {{S}tructural basis of {CDNF} interaction with the {UPR}
regulator {GRP}78},
journal = {Nature Communications},
volume = {15},
number = {1},
issn = {2041-1723},
address = {[London]},
publisher = {Nature Publishing Group UK},
reportid = {PUBDB-2024-07265},
pages = {8175},
year = {2024},
abstract = {Cerebral dopamine neurotrophic factor (CDNF) is an
unconventional neurotrophic factor that is a
disease-modifying drug candidate for Parkinson’s disease.
CDNF has pleiotropic protective effects on stressed cells,
but its mechanism of action remains incompletely understood.
Here, we use state-of-the-art advanced structural techniques
to resolve the structural basis of CDNF interaction with
GRP78, the master regulator of the unfolded protein response
(UPR) pathway. Subsequent binding studies confirm the
obtained structural model of the complex, eventually
revealing the interaction site of CDNF and GRP78. Finally,
mutating the key residues of CDNF mediating its interaction
with GRP78 not only results in impaired binding of CDNF but
also abolishes the neuroprotective activity of CDNF-derived
peptides in mesencephalic neuron cultures. These results
suggest that the molecular interaction with GRP78 mediates
the neuroprotective actions of CDNF and provide a structural
basis for development of next generation CDNF-based
therapeutic compounds against neurodegenerative diseases.},
cin = {EMBL-User / EMBL},
ddc = {500},
cid = {I:(DE-H253)EMBL-User-20120814 / I:(DE-H253)EMBL-20120731},
pnm = {6G3 - PETRA III (DESY) (POF4-6G3) / iNEXT-Discovery -
Infrastructure for transnational access and discovery in
structural biology (871037)},
pid = {G:(DE-HGF)POF4-6G3 / G:(EU-Grant)871037},
experiment = {EXP:(DE-H253)P-P12-20150101},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:39289391},
UT = {WOS:001376977000003},
doi = {10.1038/s41467-024-52478-0},
url = {https://bib-pubdb1.desy.de/record/618954},
}